Makaleler

Makale Adı Yazarlar Yayın Yeri Yılı Açıklama
1 infoEvaluation of anti-glioma effects of benzothiazoles as efficient apoptosis inducers and DNA cleaving agentsSEVER BELGİN,ÇİFTÇİ HALİLİBRAHİMMolecular and Cellular Biochemistry2023Uluslararası, Hakemli, Basılı+Elektronik, SCI-Expanded
2 infoStructural Characterization of TRAF6 N-Terminal for Therapeutic Uses and Computational Studies on New DerivativesÇİFTÇİ HALİLİBRAHİM,AYTEMİR MUTLU,DEMİRCİ HASAN,SEVER BELGİN,Fujita Mikako,Otsuka Masami,Tateishi Hiroshi,Koga Ryoko,Radwan Mohamed OPharmaceuticals2023Uluslararası, Hakemli, Basılı+Elektronik, SCI-Expanded
3 infoRapid and efficient ambient temperature X-ray crystal structure determination at Turkish Light SourceGul Mehmet,Ayan Esra,Destan Ebru,Johnson J.Austin,Shafei Alaleh,Kepceoğlu Abdullah,Yilmaz Merve,Ertem Fatma Betül,Yapici İlkin,Tosun Bilge,Baldir Nilüfer,Tokay Nurettin,Nergiz Zeliş,Karakadioğlu Gözde,Paydos Seyide Seda,Kulakman Cahine,Ferah Cengiz Kaan,Güven Ömür,Atalay Necati,Akcan Enver Kamil,Cetinok Haluk,Arslan Nazlı Eylül,Şabanoğlu Kardelen,Aşci Bengisu,Tavli Serra,Gümüsboğa Helin,Altuntaş Sevde,Otsuka Masami,Fujita Mikako,TEKİN ŞABAN,ÇİFTÇİ HALİLİBRAHİM,DURDAĞI SERDAR,KARACA EREK EZGİ,KAPLAN TÜRKÖZ BURCU,KABASAKAL BURAK VELİ,KATI AHMET,DEMİRCİ HASANScientific Reports2023Uluslararası, Hakemli, Basılı+Elektronik, SCI-Expanded
4 infoComparative Study of High-Resolution LysB29(Nε-myristoyl) des(B30) Insulin Structures Display Novel Dynamic Causal Interrelations in Monomeric-Dimeric MotionsAyan Esra,Destan Ebru,KEPCEOĞLU ABDULLAH,ÇİFTÇİ HALİLİBRAHİM,KATI AHMET,DEMİRCİ HASANCrystals2023Uluslararası, Hakemli, Basılı+Elektronik, SCI-Expanded
5 infoCryogenic X-ray crystallographic studies of biomacromolecules at Turkish Light Source <i>Turkish DeLight</i>ATALAY Necati,AKCAN Enver Kamil,GÜL Mehmet,AYAN Esra,DESTAN Ebru,ERTEM Fatma Betül,TOKAY Nurettin,ÇAKILKAYA Barış,NERGİZ Zeliş,KARAKADIOĞLU Gözde,KEPCEOĞLU ABDULLAH,YAPICI İlkin,TOSUN Bilge,BALDIR Nilüfer,YILDIRIM Günseli,JOHNSON J Austin,GÜVEN Ömür,SHAFIEI Alaleh,ARSLAN Nazlı Eylül,YILMAZ Merve,KULAKMAN Cahine,PAYDOS Seyide Seda,ÇİNAL Zeynep Sena,ŞABANOĞLU Kardelen,PAZARÇEVİREN Ayşegül,YILMAZ Ayşenur,CANBAY Başak,AŞCI Bengisu,KARTAL Esra,TAVLI Serra,ÇALISEKİ Mehmet,GÖÇ Günce,MERMER Arif,YEŞİLAY Gamze,ALTUNTAŞ Sevde,Tateishi Hiroshi,Otsuka Masami,Fujita Mikako,TEKİN ŞABAN,ÇİFTÇİ HALİLİBRAHİM,DURDAĞI SERDAR,DİNLER DOĞANAY GİZEM,KARACA EREK EZGİ,KAPLAN TÜRKÖZ BURCU,KABASAKAL BURAK VELİ,KATI AHMET,DEMİRCİ HASANTurkish Journal of Biology2023Uluslararası, Hakemli, Basılı+Elektronik, SCI-Expanded
6 infoTurkish Plants, Including Quercetin and Oenothein B, Inhibit the HIV-1 Release and Accelerate Cell ApoptosisTahara Yurika,Fujita Mikako,Otsuka Masami,Zhang Tianli,Wang Dongxing,Tateishi Hiroshi,Togami Akihiro,Nyame Perpetual,Terasawa Hiromi,Monde Nami,Appiah-Kubi Joyce,Amesimeku Wright Ofotsu,Alsaadi Doaa Husham Majeed,Wada Mikiyo,Sugimura Koji,ÇİFTÇİ HALİLİBRAHİM,GEZİCİ SEVGİ,KARAHAN FARUK,ŞEKEROĞLU NAZIM,Sawa Tomohiro,Maeda Yosuke,Watanabe Takashi,Monde KazuakiBiological and Pharmaceutical Bulletin2023Uluslararası, Hakemli, Basılı+Elektronik, SCI-Expanded
7 infoStudies on 1,4-Quinone Derivatives Exhibiting Anti-Leukemic Activity along with Anti-Colorectal and Anti-Breast Cancer EffectsÇİFTÇİ HALİLİBRAHİM,SEVER BELGİN,KAYA NUSRET,BAYRAK NİLÜFER,YILDIZ MAHMUT,YILDIRIM HATİCE,Tateishi Hiroshi,Otsuka Masami,Fujita Mikako,TUYUN AMAÇ FATİHMolecules2022Uluslararası, Hakemli, Basılı+Elektronik, SCI-Expanded
8 infoA New Series of Antileukemic Agents: Design, Synthesis, In Vitro and In Silico Evaluation of Thiazole-Based ABL1 Kinase InhibitorsZeytün Ebru,Altıntop Mehlika Dilek,SEVER BELGİN,ÖZDEMİR AHMET,Ellakwa Doha E,Ocak Zeynep,ÇİFTÇİ HALİLİBRAHİM,Otsuka Masami,Fujita Mikako,Radwan Mohamed OAnti-Cancer Agents in Medicinal Chemistry2021Uluslararası, Hakemli, Basılı+Elektronik, SCI-Expanded
9 infoIn Vitro and In Silico Evaluation of Anticancer Activity of New Indole-Based 1,3,4-Oxadiazoles as EGFR and COX-2 InhibitorsSEVER BELGİN,Altıntop Mehlika Dilek,ÖZDEMİR AHMET,AKALIN ÇİFTÇİ GÜLŞEN,Ellakwa Doha E.,Tateishi Hiroshi,Radwan Mohamed O.,Ibrahim Mahmoud A. A.,Otsuka Masami,Fujita Mikako,ÇİFTÇİ HALİLİBRAHİM,Ali Taha FSMolecules2020Uluslararası, Hakemli, Basılı+Elektronik, SCI-Expanded
10 infoStructure activity study of S-trityl-cysteamine dimethylaminopyridine derivatives as SIRT2 inhibitors: Improvement of SIRT2 binding and inhibitionRadwan Mohamed O,ÇİFTÇİ HALİLİBRAHİM,Ali Taha F.S.,Koga Ryoko,Tateishi Hiroshi,Nakata Akiko,Ito Akihiro,Yoshida Minoru,Fujita Mikako,Otsuka MasamiBioorganic & Medicinal Chemistry Letters2020Uluslararası, Hakemli, Basılı+Elektronik, SCI-Expanded
11 infoAnticancer activity of Turkish marine extracts: a purple sponge extract induces apoptosis with multitarget kinase inhibition activityÇİFTÇİ HALİLİBRAHİM,CAN MUSTAFA,Ellakwa Doha E,Suner Salih C,Ibrahim Mohamed A,ORAL AYHAN,ŞEKEROĞLU NAZIM,ÖZALP HASAN BARIŞ,Otsuka Masami,Fujita Mikako,ALPARSLAN MUSTAFA,O Radwan MohamedInvestigational New Drugs2020Uluslararası, Hakemli, Basılı+Elektronik, SCI-Expanded
12Antiproliferative Activity of α-Tomatine and Molecular Target IdentificationÇİFTÇİ HALİLİBRAHİMTürk Tarım ve Doğa Bilimleri Dergisi2020Ulusal, Hakemli, Elektronik, TR DİZİN
13 infoEffects of Glycyrrhetic Acid on Human Chronic Myelogenous Leukemia CellsÇİFTÇİ HALİLİBRAHİMTurkish Journal of Pharmaceutical Sciences2020Uluslararası, Hakemli, Elektronik, ESCI
14 infoA novel series of chlorinated plastoquinone analogs: Design, synthesis, and evaluation of anticancer activityBayrak Nilufer,YILDIRIM HATİCE,YILDIZ MAHMUT,Radwan Mohamed O,Otsuka Masami,Fujita Mikako,ÇİFTÇİ HALİLİBRAHİM,Tuyun Amac FatihChemical Biology Drug Design2020Uluslararası, Hakemli, Elektronik, SCI
15 infoAntileukemic Activity of Twig Components of Caucasian Beech in TurkeyShida Wataru,Tateishi Hiroshi,Tahara Yurika,Fujita Mikako,Doaa Husam Majeed Alsaadi,Masato Watanabe,Koga Ryoko,Radwan Mohamed O,ÇİFTÇİ HALİLİBRAHİM,GEZİCİ SEVGİ,Kuraichi Yuki,Katsuki Hiroshi,Otsuka Masami,Sugimura Koji,Wada Mikiyo,Sekeroglu Nazim,Watanabe TakashiMolecules2019Uluslararası, Hakemli, Elektronik, SCI-Expanded
16 infoDesign, synthesis and biological evaluation of a new series of thiazolyl-pyrazolines as dual EGFR and HER2 inhibitorsSEVER BELGİN,Altıntop Mehlika Dilek,Radwan Mohamed O,ÖZDEMİR AHMET,Otsuka Masami,Fujita Mikako,ÇİFTÇİ HALİLİBRAHİMEuropean Journal of Medicinal Chemistry2019Uluslararası, Hakemli, Elektronik, SCI
17 infoDiscovery and structure–activity relationship of plastoquinone analogs as anticancer agents against chronic myelogenous leukemia cellsÇİFTÇİ HALİLİBRAHİM,Bayrak Nilufer,YILDIRIM HATİCE,YILDIZ MAHMUT,Radwan Mohamed O,Otsuka Masami,Fujita Mikako,Tuyun Amac FatihArchiv der Pharmazie2019Uluslararası, Hakemli, Elektronik, SCI
18 infoDesign, synthesis, and biological activity of Plastoquinone analogs as a new class of anticancer agentsBayrak Nilufer,YILDIRIM HATİCE,YILDIZ MAHMUT,Radwan Mohamed O,Otsuka Masami,Fujita Mikako,Tuyun Amac Fatih,ÇİFTÇİ HALİLİBRAHİMBioorganic Chemistry2019Uluslararası, Hakemli, Elektronik, SCI
19 infoDesign, Synthesis and Biological Evaluation of Pentacyclic Triterpene Derivatives: Optimization of Anti-ABL Kinase ActivityÇİFTÇİ HALİLİBRAHİM,Radwan Mohamed O,Ozturk Safiye Emirdag,Ulusoy N Gokce,Ece Sozer,Ellakwa Doha E,Ocak Zeynep,Can Mustafa,Ali Taha FS,AbdAlla Howaida I,Yayli Nurettin,Tateishi Hiroshi,Otsuka Masami,Fujita MikakoMolecules2019Uluslararası, Hakemli, Elektronik, SCI-Expanded
20 infoSerial Femtosecond X-Ray Diffraction of HIV-1 Gag MA-IP6 Microcrystals at Ambient TemperatureÇİFTÇİ HALİLİBRAHİM,Sierra Raymond G,Yoon Chun Hong,Zhen Su,Tateishi Hiroshi,Koga Ryoko,Kotaro Koiwai,Yumoto Fumiaki,Senda Toshiya,Liang Meng,Soichi Wakatsuki,Otsuka Masami,Fujita Mikako,DeMirci HasanInternational Journal of Molecular Sciences2019Uluslararası, Hakemli, Elektronik, SCI-Expanded
21 infoAntiproliferative S-Trityl-l-Cysteine -Derived Compounds as SIRT2 Inhibitors: Repurposing and Solubility EnhancementRadwan Mohamed O,ÇİFTÇİ HALİLİBRAHİM,Ali Taha FS,Ellakwa Doha E,Koga Ryoko,Tateishi Hiroshi,Nakata Akiko,Ito Akihori,Minoru Yoshida,Okamoto Yoshinari,Fujita Mikako,Otsuka MasamiMolecules2019Uluslararası, Hakemli, Elektronik, SCI-Expanded
22 infoNew SIRT2 inhibitors: Histidine-based bleomycin spin-offAli Taha FS,ÇİFTÇİ HALİLİBRAHİM,Radwan Mohamed O,Koga Ryoko,Ohsugi Takeo,Okiyama Yoshio,Teruki Honma,Nakata Akiko,Ito Akihori,Minoru Yoshida,Fujita Mikako,Otsuka MasamiBioorganic Medicinal Chemistry2019Uluslararası, Hakemli, Elektronik, SCI
23 infoDesign, Synthesis, and Biological Evaluation of Novel 1,3,4-Thiadiazole Derivatives as Potential Antitumor Agents against Chronic Myelogenous Leukemia: Striking Effect of Nitrothiazole MoietyAltıntop Mehlika Dilek,ÇİFTÇİ HALİLİBRAHİM,Radwan Mohamed O,SEVER BELGİN,KAPLANCIKLI ZAFER ASIM,Ali Taha FS,Koga Ryoko,Fujita Mikako,Otsuka Masami,ÖZDEMİR AHMETMolecules2018Uluslararası, Hakemli, Elektronik, SCI-Expanded
24 infoAminoglycoside ribosome interactions reveal novel conformational states at ambient temperatureMary E OSullivan,Poitevin Frederic,Sierra Raymond G,Gati Cornelius,Dao E Han,Rao Yashas,Aksit Fulya,ÇİFTÇİ HALİLİBRAHİM,Corsepius Nicholas,Robert Greenhouse,Hayes Matt J,Hunter Mark S,Liang Meng,Alex McGurk,Paul Mgbam,Obrinski Trevor,Fatima PardoAvila,Seaberg Matt,Cheng Alan G,Ricci Anthony J,DeMirci HasanNucleic Acids Research2018Uluslararası, Hakemli, Elektronik, SCI
25 infoStructure of the 30S ribosomal decoding complex at ambient temperatureDao E Han,Poitevin Frederic,Sierra Raymond G,Gati Cornelius,Rao Yashas,ÇİFTÇİ HALİLİBRAHİM,Aksit Fulya,Alex McGurk,Obrinski Trevor,Mgbam Paul,Hayes Matt J,Lichtenberg Casper de,Fatima PardoAvila,Corsepius Nicholas,Zhang Lindsey,Seaberg Matt,Hunter Mark S,Liang Meng,Koglin Jason E,Soichi Wakatsuki,DeMirci HasanRNA2018Uluslararası, Hakemli, Elektronik, SCI
26 infoIntroduction of H2C2-type zinc-binding residues into HIV-2 Vpr increases its expression levelKoga Ryoko,Yamamoto Minami,ÇİFTÇİ HALİLİBRAHİM,Otsuka Masami,Fujita MikakoFEBS Open Bio2018Uluslararası, Hakemli, Elektronik, SCI-Expanded
27 infoThe First Pentacyclic Triterpenoid Gypsogenin Derivative Exhibiting Anti-ABL1 Kinase and Anti-chronic Myelogenous Leukemia ActivitiesÇİFTÇİ HALİLİBRAHİM,Ozturk Safiye Emirdag,Ali Taha FS,Radwan Mohamed O,Tateishi Hiroshi,Koga Ryoko,Ocak Zeynep,Can Mustafa,Otsuka Masami,Fujita MikakoBiological and Pharmaceutical Bulletin2018Uluslararası, Hakemli, Elektronik, SCI
28 infoSe-SAD serial femtosecond crystallography datasets from selenobiotinyl-streptavidinYoon Chun Hong,DeMirci Hasan,Sierra Raymond G,Dao E Han,Ahmadi Radman,Aksit Fulya,Aquila Andrew L,Alexander Batyuk,ÇİFTÇİ HALİLİBRAHİM,Guillet Serge,Hayes Matt J,Lane Thomas J,Liang Meng,Lundström Ulf,Koglin Jason E,Mgbam Paul,Rao Yashas,Rendahl Theodore,Rodriguez Evan,Zhang Lindsey,Soichi Wakatsuki,Boutet Sbastien,James M Holton,Hunter Mark SScientific Data2017Uluslararası, Hakemli, Elektronik, SCI-Expanded
29 infoZinc-binding site of human immunodeficiency virus 2 Vpx prevents instability and dysfunction of the proteinYamamoto Minami,Koga Ryoko,Fujino Haruna,Shimagaki Kazunori,ÇİFTÇİ HALİLİBRAHİM,Kamo Masahiro,Tateishi Hiroshi,Otsuka Masami,Fujita MikakoJournal of General Virology2017Uluslararası, Hakemli, Elektronik, SCI
30 infoA Dithiol Compound Binds to the Zinc Finger Protein TRAF6 and Suppresses Its UbiquitinationKoga Ryoko,Radwan Mohamed O,Ejima Tomohiko,Kanemaru Yosuke,Tateishi Hiroshi,Ali Taha FS,ÇİFTÇİ HALİLİBRAHİM,Shibata Yuri,Yuu Taguchi,Inoue Junichiro,Otsuka Masami,Fujita MikakoChemMedChem2017Uluslararası, Hakemli, Elektronik, SCI
31 infoA clue to unprecedented strategy to HIV eradication: “Lock-in and apoptosis”Tateishi Hiroshi,Monde Kazuaki,Anraku Kensaku,Koga Ryoko,Hayashi Yuya,ÇİFTÇİ HALİLİBRAHİM,DeMirci Hasan,Higashi Taishi,Keiichi Motoyama,Arima Hidetoshi,Otsuka Masami,Fujita MikakoScientific Reports2017Uluslararası, Hakemli, Elektronik, SCI
32 infoSynthesis, Computational Study, and Evaluation of in vitro Antimicrobial, Antibiofilm, and Anticancer Activities of New Sulfanyl Aminonaphthoquinone DerivativesBayrak Nilufer,YILDIRIM HATİCE,Tuyun Amac Fatih,Kara Emel Mataraci,Celik Berna Ozbek,Gupta Girish Kumar,ÇİFTÇİ HALİLİBRAHİM,Fujita Mikako,Otsuka Masami,Nasiri Hamid RLetters in Drug Design Discovery2017Uluslararası, Hakemli, Elektronik, SCI-Expanded
33 infoSelenium single-wavelength anomalous diffraction de novo phasing using an X-ray-free electron laserHunter Mark S,Yoon Chun Hong,DeMirci Hasan,Sierra Raymond G,Dao E Han,Ahmadi Radman,Aksit Fulya,Aquila Andrew L,ÇİFTÇİ HALİLİBRAHİM,Guillet Serge,Hayes Matt J,Lane Thomas J,Liang Meng,Lundström Ulf,Koglin Jason E,Paul Mgbam,Yashas Rao,Zhang Lindsey,Soichi Wakatsuki,James M Holton,Boutet SbastienNature Communications2016Uluslararası, Hakemli, Elektronik, SCI
34 infoNovel metal chelating molecules with anticancer activity. Striking effect of the imidazole substitution of the histidine–pyridine–histidine systemAli Taha FS,Iwamaru Kana,ÇİFTÇİ HALİLİBRAHİM,Koga Ryoko,Matsumoto Masahiro,Oba Yasunori,Hiromasa Kurosaki,Fujita Mikako,Okamoto Yoshinari,Umezawa Kazuo,Nakao Mitsuyoshi,Hide Takuichiro,Makino Keishi,Kuratsu Junichi,AbdelAziz Mohamed,Gamal ElDin AA AbuoRahma,Eman AM Beshr,Otsuka MasamiBioorganic Medicinal Chemistry2015Uluslararası, Hakemli, Elektronik, SCI
35 infoSynthesis and Evaluation of New Pyrazoline Derivatives as Potential Anticancer AgentsKarabacak Muhammed,Altıntop Mehlika Dilek,ÇİFTÇİ HALİLİBRAHİM,Koga Ryoko,Otsuka Masami,Fujita Mikako,ÖZDEMİR AHMETMolecules2015Uluslararası, Hakemli, Elektronik, SCI-Expanded
36 infoMutational analysis of HIV-2 Vpx shows that proline residue 109 in the poly-proline motif regulates degradation of SAMHD1ÇİFTÇİ HALİLİBRAHİM,Fujino Haruna,Koga Ryoko,Yamamoto Minami,Kawamura Sogo,Tateishi Hiroshi,Yasumasa Iwatani,Otsuka Masami,Fujita MikakoFEBS Letters2015Uluslararası, Hakemli, Elektronik, SCI